Relugolix 737789-87-6 pharmaceutical intermediate

Basic Chemical Information

Product Introduction

Relugolix (aliases TAK-385, RVT-601) is a highly specific fluorinated heterocyclic small-molecule organic compound, serving as a dedicated research substrate for in vitro endocrine receptor mechanism studies. It features a stable molecular skeleton, regular functional group distribution and strong spatial structure specificity, with excellent chemical structural stability and degradation resistance. The material presents pure and uniform texture under normal conditions without structural defects. It is not prone to oxidation, discoloration or deliquescence at room temperature, maintaining complete molecular skeleton and inherent biological affinity during long-term storage.As a core experimental material in the field of gonadotropin-releasing hormone receptor research, this molecule has highly specific target-binding properties and wide substrate adaptability, stably applicable to various in vitro biochemical research systems at molecular and cellular levels with excellent repeatability.

Application Scope 

GnRH Receptor Mechanism Research： As a typical GnRH receptor antagonist small molecule, it is stably applied to in vitro receptor binding assays, target affinity detection and receptor signaling pathway blocking mechanism analysis. Featuring high action specificity and no off-target interference, it delivers highly repeatable experimental data and serves as a core tool compound for basic endocrine receptor research.

Endocrine and Reproductive Signal Regulation Research： It is used to explore the secretion regulation mechanism of luteinizing hormone and follicle-stimulating hormone in in vitro cell models, suitable for basic research on sex hormone signaling pathways and endocrine homeostasis regulation, and widely applied in in vitro mechanism verification of reproductive and endocrine pharmacology.

Organic Synthesis & Structural Derivation R&D： With multiple active functional groups including fluorinated benzyl, thiophene ring and urea groups, it features strong structural plasticity. As a core synthetic intermediate, it supports structural modification, group decoration, lead compound screening and structure-activity relationship research for new GnRH antagonist heterocyclic derivatives.

Academic Experiment Reproduction & System Control： Its physicochemical properties are fully consistent with international standard research-grade materials, enabling accurate reproduction of published in vitro molecular experiments, cell activity tests and target inhibition gradient assays for academic research deepening, experimental system calibration and research data verification.

Molecular Structural Stability Special Research： Based on its excellent structural stability, it supports research on molecular structural evolution and functional group degradation rules under light, temperature fluctuation and acid-base solvent systems for special research on small-molecule compound physicochemical properties and structural stability.

Important Disclaimer

This product is an organic chemical intermediate for pure scientific research, only used as laboratory chemical material. It is not drug, veterinary drug, health product, food or cosmetic raw material with no medical, commercial or civilian value and no therapeutic or health-care effects. Purchasers confirm the purpose of formal laboratory scientific research and promise not to change the use. All risks and legal liabilities arising from illegal misappropriation and abuse shall be borne independently by purchasers.

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